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UNMC Researchers First in United States to Begin Study on Safety, Effectiveness of Unique New Drug for Potential Treatment of Acute Myeloid Leukemia (AML)

University of Nebraska Medical Center researchers have begun the first

clinical study in the United States to examine the safety and effectiveness

of a unique new drug that may have potential in the treatment of acute

myeloid leukemia (AML). AML, a cancer of the blood and bone marrow, is

the most common type of acute leukemia in adults, with an estimated 10,000

new cases a year.

UNMC is conducting the first and second phase of a clinical study in

adults, age 19 and over, whose treatment has failed or whom are not eligible

for conventional chemotherapy. Those who have not yet received any treatment

for their disease also may be considered for the study.

The goal of the study is to evaluate how safe the drug is and how effective

it is in inhibiting the growth of leukemia cells.

Participants will receive treatment at no extra cost on an outpatient

basis in the Lied Transplant Center on the UNMC/NHS campus. Study participants

will receive the drug on an outpatient basis. Participants can be part

of the study and continue to see their own physicians. They may refer themselves

or be referred to UNMC by their physicians.

James Foran, M.D., principal investigator of the UNMC study, said the

oral drug, whose name is currently confidential because of proprietary

issues, is part of a new class of drugs called receptor tyrosine kinases

(RTK) inhibitors, which appear to play an important role in the disease

process. He said the drug might be a potential adjunct, or additional treatment,

in what frequently is an incurable disease.

Leukemia cells in most patients express RTKs, or growth receptors, which,

when interacting with their respective growth factors, cause leukemia cells

to multiply.

There is no standard therapy for those whose initial treatment has

failed or are not eligible for conventional chemotherapy. Even with any

successive standard therapy, prognosis is poor, with an average survival

in the range of three months, said Dr. Foran, an oncologist and assistant

professor at UNMC.

This is a new treatment approach to leukemia. Initial studies in healthy

volunteers suggest that single doses of the drug are well-tolerated, and

about a dozen patients are currently being treated with this medication

for other cancer, in Europe and the United States, Dr. Foran said. This

is the first study in leukemia, and it is a very exciting opportunity at

UNMC to improve our understanding of how leukemia cells survive, how we

can bypass those survival mechanisms, and ultimately develop better treatments

for this disease.

The study is funded by Sugen, Inc., now part of Pharmacia Corporation,

a worldwide pharmaceutical company. Dr. Foran said UNMC was the first site

chosen to test the drug in AML because of its cancer research and clinical

programs.

 Dr. Foran said studies like this enable researchers to learn more

about the biology of the disease in order to design new treatments with

better results and fewer side effects.

There are major changes, astonishing developments in our approach to

the treatment of cancer. This is due to research and the different way

we are thinking about and targeting cancers specifically. The changes Ive

seen in 10 years are incredible, he said.

Drugs like this are changing the way we think about leukemia, and I

believe will change the way we treat leukemia in the next few years, Dr.

Foran said. We probably wont get rid of chemotherapy because of its

effectiveness, but drugs like these will be important additions to therapy.

The Leukemia and Lymphoma Society estimates about 21,500 deaths in the

U.S. in 2001 resulted from leukemia. Of that, about one-third (7,200) died

from acute myelogenous leukemia.

AML, a rapidly progressing disease that originates in a cell in the

marrow, causes uncontrolled growth of developing marrow cells that affect

the body’s ability to fight infections. Dr. Foran said about one in four

patients under 60 years old with AML can be cured, but the disease in those

60 and over is much more difficult to cure.

AML is the most common form of acute leukemia and occurs mostly in people

in their 60s, 70s and 80s. The cause is unknown in most cases.

UNMC/NHS is recognized internationally for its expertise in the diagnosis

and treatment of leukemias and lymphomas and is one of the busiest bone

marrow and stem cell transplant centers in the world. James Armitage, M.D.,

now dean of the UNMC College of Medicine, launched the program in 1982.

Other physicians working on the study are UNMC oncologists Phil Bierman,

M.D., Gregory Bociek, M.D., Anne Kessinger, M.D., Steven Pavletic, M.D.,

Elizabeth Reed, M.D., Stefano Tarantolo, M.D. and Julie Vose, M.D.

For more information about the study, call Maribeth Hohenstein at (402)

559-9053.